Found 58 of ec50 for Adrenergic receptor alpha-2
having polymerids = 49000232 and
complexids = 50000720,50003305
having polymerids = 49000232 and
complexids = 50000720,50003305
Affinity DataEC50: 41nMAssay Description:Effective Concentration at Alpha-2B adrenergic receptor from CHO-RNG cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Effective Concentration at Alpha-2B adrenergic receptor from CHO-RNG cellsMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonistic potency at beta-1 adrenergic receptor for the percent maximal increase in contraction rate of isolated guinea pig atriaMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 166nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonistic potency at alpha 2-Adrenergic receptor for inhibition of 10 uM forskolin-elicited stimulation of adenylate cyclase in human platelet membra...More data for this Ligand-Target Pair
Affinity DataEC50: 470nMAssay Description:Effective Concentration at Alpha-2B adrenergic receptor from CHO-RNG cellsMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Activity at alpha2 adrenergic receptor in human brain prefrontal cortex membranes assessed as effect on UK14304-induced [35S]GTPgammaS binding by mea...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Activity at alpha2 adrenergic receptor in human brain prefrontal cortex membranes assessed as effect on UK14304-induced [35S]GTPgammaS binding by mea...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Effective Concentration at Alpha-2B adrenergic receptor from CHO-RNG cellsMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Effective concentration (EC50) against alpha-2-adrenoceptor in the guinea pig atriumMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Activity at alpha2 adrenergic receptor in human brain prefrontal cortex membranes assessed as effect on UK14304-induced [35S]GTPgammaS binding by mea...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Activity at alpha2 adrenergic receptor in human brain prefrontal cortex membranes assessed as effect on UK14304-induced [35S]GTPgammaS binding by mea...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at alpha2 adrenoceptor in human cortical membrane after 2 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 2.71E+3nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 2.76E+3nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 3.57E+3nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 4.14E+3nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 4.23E+3nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 4.38E+3nMAssay Description:Antagonist activity at human brain adrenergic alpha-2 receptor assessed as UK-14304-stimulated [35S]GTPgammaS binding at 10 uMMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic potency at alpha 2-Adrenergic receptor for inhibition of 10 uM forskolin-elicited stimulation of adenylate cyclase in human platelet membra...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 6.60E+3nMAssay Description:Activity at alpha2 adrenergic receptor in human brain prefrontal cortex membranes assessed as effect on UK14304-induced [35S]GTPgammaS binding by mea...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 6.71E+3nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.02E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.07E+4nMAssay Description:Activity at alpha2 adrenergic receptor in human brain prefrontal cortex membranes assessed as effect on UK14304-induced [35S]GTPgammaS binding by mea...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.14E+4nMAssay Description:Activity at alpha2 adrenergic receptor in human brain prefrontal cortex membranes assessed as effect on UK14304-induced [35S]GTPgammaS binding by mea...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.14E+4nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.14E+4nMAssay Description:Agonist activity at alpha2 adrenoceptor in human cortical membrane after 2 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.16E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.60E+4nMAssay Description:Antagonist activity at human brain adrenergic alpha-2 receptor assessed as UK-14304-stimulated [35S]GTPgammaS binding at 10 uMMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.62E+4nMAssay Description:Agonist activity at alpha2 adrenoceptor in human cortical membrane after 2 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.80E+4nMAssay Description:Agonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation spe...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 2.02E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 3.00E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 3.04E+4nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 3.08E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 3.70E+4nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 3.87E+4nMAssay Description:Agonist activity at alpha2 adrenoceptor in human cortical membrane after 2 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 3.99E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 4.22E+4nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 4.53E+4nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 4.60E+4nMAssay Description:Agonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation spe...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 5.23E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 5.64E+4nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 5.93E+4nMAssay Description:Agonist activity at alpha2 adrenoceptor in human cortical membrane after 2 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 6.03E+4nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 6.14E+4nMAssay Description:Agonist activity at alpha2 adrenoceptor in human cortical membrane after 2 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 8.23E+4nMAssay Description:Agonist activity at alpha2 adrenoceptor in human cortical membrane after 2 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 8.72E+4nMAssay Description:Antagonist activity at adrenergic alpha 2 receptor in human brain membrane assessed as inhibition of UK14304-induced stimulation of [35S]GTPgammaS bi...More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.20E+5nMAssay Description:Agonist activity at human brain adrenergic alpha2 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataEC50: 1.41E+5nMAssay Description:Antagonist activity at human brain adrenergic alpha-2 receptor assessed as UK-14304-stimulated [35S]GTPgammaS binding at 10 uMMore data for this Ligand-Target Pair